KT5823 for cell activation

Catalog number
2164-50
Name
KT5823 for cell activation
Size
50 µg
Price
159.00 EUR
Supplier

Details

Description
Cell-permeable. KT5823 is a derivative of K-252a (Cat. No. 2013) that acts as a selective inhibitor of Protein kinase G (PKG) (Ki = 0.234 µM). Inhibits other kinases at much higher concentrations (Ki’s for PKA = 4 μM and for MLCK=>10 μM).
Peptide sequence
N/A
CAS number
126643-37-6
Molecular weight
495.53
Category
Biochemicals
Other name
2,​3,​9,​10,​11,​12-​hexahydro-​10R-​methoxy-​2,​9-​dimethyl-​1-​oxo-​ 9S,​12R-​epoxy-​1H-​diindolo[1,​2,​3-​fg:3’,​2’,​1’-​kl]pyrrolo[3,​4-​ i][1,​]benzodiazocine-​10-​carboxylic acid,​ methyl ester
Molecular formula
C₂₉H₂₅N₃O₅
Physical appearance
White solid
Supplied with
N/A
Is this a salt?
No
Is it cell-permeable?
Yes
Purification
≥98% by HPLC
Reconstitute instructions
DMSO (20 mg/ml)
Storage condition
-20°C
Shipping condition
gel pack
Maximum time for storage
24months
Storage instructions
Protect from air and light
Tissue
cell
Additional description
For cells, cell lines and tissues in culture till half confluency.