PFI-1 for cell activation

Catalog number
2203-1
Name
PFI-1 for cell activation
Size
1 mg
Price
115.00 EUR
Supplier

Details

Description
PFI-1 is a BET bromodomain inhibitor that exhibits inhibitory activity at BRD2 and BRD4. In an AlphaScreen assay it has been shown to inhibit BRD2 bromodomain 2 and BRD4 bromodomain 1 with IC₅₀ values of 98 nM and 0.22 μM, respectively.
Peptide sequence
N/A
CAS number
N/A
Molecular weight
347.39
Category
Biochemicals
Other name
2-​Methoxy-​N-​(3-​methyl-​2-​oxo-​1,​2,​3,​4-​tetrahydroquinazolin-​6-​yl)benzenesulfonamide
Molecular formula
C₁₆H₁₇N₃O₄S
Physical appearance
Beige solid
Supplied with
N/A
Is this a salt?
No
Is it cell-permeable?
Yes
Purification
≥98%
Reconstitute instructions
DMSO (50 mM)
Storage condition
-20°C
Shipping condition
gel pack
Maximum time for storage
24months
Storage instructions
Protect from air and light
Tissue
cell
Additional description
For cells, cell lines and tissues in culture till half confluency.