Enzastaurin (LY317615) for cell activation

Catalog number
1619-1
Name
Enzastaurin (LY317615) for cell activation
Size
1 mg
Price
219.00 EUR
Supplier

Details

Description
Enzastaurin (Enz) is a potent and selective inhibitor of PKCβ with antiproliferative activity (IC₅₀= ~6 nM). Enz suppresses VEGF-induced angiogenesis in the rat corneal micropocket assay, decreases microvessel density, and prevents VEGF secretion from human tumor cell xenografts in nude mice. Prolonged courses of Enz increase chemotherapy or radiation tumor growth delay of glioma, breast, and small cell lung cancer xenografts.
Peptide sequence
N/A
CAS number
170364-57-5
Molecular weight
515.61
Category
Biochemicals
Other name
LY317615, LY-317615, D04014
Molecular formula
C₃₂H₂₉N₅O₂
Physical appearance
Red-Orange Solid
Supplied with
N/A
Is this a salt?
No
Is it cell-permeable?
Yes
Purification
≥99% by HPLC
Reconstitute instructions
DMSO (5 mg/ml)
Storage condition
-20°C
Shipping condition
RT
Maximum time for storage
24months
Storage instructions
Protect from air and light
Tissue
cell
Additional description
For cells, cell lines and tissues in culture till half confluency.