TGX-221 for cell activation
Catalog number
1781-1
Name
TGX-221 for cell activation
Size
1 mg
Price
148.00 EUR
Supplier
Details
Description
Cell-permeable. A potent, selective and ATP-competitive inhibitor of PI 3-kinase β (IC₅₀ = 5 nM for p110β). Inhibits other PI3K isoforms at higher concentrations (IC₅₀ = 0.1 µM for p110δ, 5 µM for p110⍺, and 3.5 µM for p110ɣ).
Peptide sequence
N/A
CAS number
663619-89-4
Molecular weight
364.44
Category
Biochemicals
Other name
(±)-7-Methyl-2-(morpholin-4-yl)-9-(1-phenylaminoethyl)-pyrido[1,2-a]-pyrimidin-4-one
Molecular formula
C₂₁H₂₄N₄O₂
Physical appearance
White solid
Supplied with
N/A
Is this a salt?
No
Is it cell-permeable?
Yes
Purification
≥98% by HPLC
Reconstitute instructions
DMSO (10 mg/ml) or Ethanol (5 mg/ml)
Storage condition
-20°C
Shipping condition
gel pack
Maximum time for storage
48 months
Storage instructions
Protect from air and light
Tissue
cell
Additional description
For cells, cell lines and tissues in culture till half confluency.
