KT5720 for cell activation

Catalog number
2276-100
Name
KT5720 for cell activation
Size
100 µg
Price
306.00 EUR
Supplier

Details

Description
A derivative of the protein kinase inhibitor K252a (Cat. No. 2013). Acts as a potent, selective, ATP-competitive inhibitor of protein kinase A (PKA) (Ki = 60 nM). Has no effect on PKC, PKG and MLCK.
Peptide sequence
N/A
CAS number
108068-98-0
Molecular weight
537.61
Category
Biochemicals
Other name
(9R,10S,12S)-2,3,9,10,11,12-Hexahyd­ro-10-hydroxy-9-methyl-1-oxo-9,12-epoxy-1H-diindol­o[1,2,3-fg:3',2',1'-kl]pyrrolo[3,4-i][1,6]benzodiazoc­ine-10-carboxylic acid, hexyl ester
Molecular formula
C₃₂H₃₁N₃O₅
Physical appearance
Colorless solid
Supplied with
N/A
Is this a salt?
No
Is it cell-permeable?
Yes
Purification
≥98% by HPLC
Reconstitute instructions
DMSO (~50 mM)
Storage condition
-20 ̊C
Shipping condition
gel pack
Maximum time for storage
24 months
Storage instructions
Protect from air and moisture
Tissue
cell
Additional description
For cells, cell lines and tissues in culture till half confluency.