GSK-3787 for cell activation

Catalog number
2400-5
Name
GSK-3787 for cell activation
Size
5 mg
Price
153.00 EUR
Supplier

Details

Description
GSK-3787 is a selective and irreversible antagonist of the peroxisome proliferator-activated receptor delta (PPARδ) (plC₅₀ = 6.6). It covalently binds to Cys 249 in the PPARδ binding site.
Peptide sequence
N/A
CAS number
188591-46-0
Molecular weight
392.78
Category
Biochemicals
Other name
4-Chloro-N-(2-{[5-(trifluoromethyl)-2-pyridyl]sulfonyl}ethyl)benzamide
Molecular formula
C₁₅H₁₂ClF₃N₂O₃S
Physical appearance
White solid
Supplied with
N/A
Is this a salt?
No
Is it cell-permeable?
Yes
Purification
≥98% by TLC
Reconstitute instructions
DMSO (~30 mg/ml)
Storage condition
-20 ̊C
Shipping condition
gel pack
Maximum time for storage
36 months
Storage instructions
Protect from light and air
Tissue
cell
Additional description
For cells, cell lines and tissues in culture till half confluency.