A-803467 for cell activation
Catalog number
2559-5
Name
A-803467 for cell activation
Size
5 mg
Price
132.00 EUR
Supplier
Details
Description
A-803467 is a potent, selective inhibitor of the TTX-resistant voltage-gated sodium channel Na(v1.8). Na(v1.8) is preferentially expressed in sensory neurons, and inhibition attenuates both inflammatory and neuropathic pain in a variety of animal models. IC50's for rat and human Na(v1.8) are 140 nM and 8.0 nM respectively.
Peptide sequence
N/A
CAS number
944261-74-9
Molecular weight
357.8
Category
Biochemicals
Other name
5-(4-Chlorophenyl)-N-(3,5-dimethoxyphenyl)furan-2-carboxamide
Molecular formula
C₁₉H₁₆ClNO₄
Physical appearance
Off-white solid
Supplied with
N/A
Is this a salt?
No
Is it cell-permeable?
Yes
Purification
≥98% by TLC
Reconstitute instructions
DMSO (~30 mg/ml) or EtOH (~ 5 mg/ml)
Storage condition
-20°C
Shipping condition
Gel pack
Maximum time for storage
24 months
Storage instructions
Protect from air and light
Tissue
cell
Additional description
For cells, cell lines and tissues in culture till half confluency.