CX-6258 for cell activation
Catalog number
2851-5
Name
CX-6258 for cell activation
Size
5 mg
Price
153.00 EUR
Supplier
Details
Description
CX-6258 is a potent pan-Pim kinases inhibitor (IC₅₀ values of 5 nM, 25 nM and 16 nM for Pim-1, Pim-2 and Pim-3, respectively). CX-6258 exhibits in vitro synergy with chemotherapeutics and robust in vivo efficacy in two Pim kinases driven tumor models.
Peptide sequence
N/A
CAS number
1202916-90-2
Molecular weight
461.94
Category
Biochemicals
Other name
(E)-5-chloro-3-((5-(3-(4-methyl-1,4-diazepane-1-carbonyl)phenyl)furan-2-yl)methylene)indolin-2-one
Molecular formula
C₂₆H₂₄ClN₃O₃
Physical appearance
White solid
Supplied with
N/A
Is this a salt?
No
Is it cell-permeable?
Yes
Purification
≥98% by HPLC
Reconstitute instructions
DMSO (>5 mg/ml)
Storage condition
-20°C
Shipping condition
gel pack
Maximum time for storage
36 months
Storage instructions
Protect from air and light
Tissue
cell
Additional description
For cells, cell lines and tissues in culture till half confluency.
