XL-147 for cell activation

Catalog number
9401-5
Name
XL-147 for cell activation
Size
5 mg
Price
229.00 EUR
Supplier

Details

Description
XL-147 is an ATP-competitive, highly selective, and reversible pan-class I phosphoinositide 3-kinase (PI3K) inhibitor. It inhibits PI3K p110α, -β, -γ, and -δ isoforms, with IC₅₀ values of 48, 617, 10, and 260 nmol/L, respectively, measured in biochemical assays. XL-147 displays antitumor activity.
Peptide sequence
N/A
CAS number
956958-53-5
Molecular weight
448.52
Category
Biochemicals
Other name
N-[3-(2,1,3-benzothiadiazol-5-ylamino)quinoxalin-2-yl]-4-methylbenzenesulfonamide; SAR245408; Pilaralisib
Molecular formula
C₂₁H₁₆N₆O₂S₂
Physical appearance
Off-white solid
Supplied with
N/A
Is this a salt?
No
Is it cell-permeable?
Yes
Purification
≥98% by HPLC
Reconstitute instructions
DMSO (~ 3 mg/ml)
Storage condition
-20°C
Shipping condition
gel pack
Maximum time for storage
36 months
Storage instructions
Protect from air and light
Tissue
cell
Additional description
For cells, cell lines and tissues in culture till half confluency.