Cobicistat for cell activation

Catalog number

9474-25

Size

25 mg

Price

643.00 EUR

Supplier

Biovision

Order

Details

Description

Cobicistat (GS-9350) is a potent, and selective inhibitor of human cytochrome P450 3A (CYP3A) enzymes (Ki = 939 nM). Acts as a pharmacoenhancing or "boosting" agent for antiviral drugs used in the treatment of HIV infection.

Peptide sequence

N/A

CAS number

1004316-88-4

Molecular weight

776.02

Category

Biochemicals

Other name

1,3-thiazol-5-ylmethyl N-[(2R,5R)-5-[[(2S)-2-[[methyl-[(2-propan-2-yl-1,3-thiazol-4-yl)methyl]carbamoyl]amino]-4-morpholin-4-ylbutanoyl]amino]-1,6-diphenylhexan-2-yl]carbamate; GS-9350

Molecular formula

C₄₀H₅₃N₇O₅S₂

Physical appearance

White to off-white solid

Supplied with

N/A

Is this a salt?

N/A

Is it cell-permeable?

Yes

Purification

≥98% by HPLC