GDC-0032 for cell activation

Catalog number
9573-25
Name
GDC-0032 for cell activation
Size
25 mg
Price
588.00 EUR
Supplier

Details

Description
GDC-0032 is a potent, and selective inhibitor of Class I PI3-K α, δ, and γ isoforms, with 30-fold less inhibition of the PI3K β isoform relative to the PI3K α isoform. This next generation PI3-K inhibitor displays increased anti-tumor activity against PIK3CA mutant (MT) cell lines.
Peptide sequence
N/A
CAS number
1282512-48-4
Molecular weight
460.53
Category
Biochemicals
Other name
2-methyl-2-[4-[2-(5-methyl-2-propan-2-yl-1,2,4-triazol-3-yl)-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl]pyrazol-1-yl]propanamide; Taselisib
Molecular formula
C₂₄H₂₈N₈O₂
Physical appearance
White to off-white solid
Supplied with
N/A
Is this a salt?
No
Is it cell-permeable?
Yes
Purification
≥98% by HPLC
Reconstitute instructions
DMSO (>10 mg/ml)
Storage condition
-20°C
Shipping condition
gel pack
Maximum time for storage
36 months
Storage instructions
Protect from air and light
Tissue
cell
Additional description
For cells, cell lines and tissues in culture till half confluency.