UNC0379 for cell activation
Catalog number
9588-5
Name
UNC0379 for cell activation
Size
5 mg
Price
186.00 EUR
Supplier
Details
Description
UNC0379 is a selective, substrate-competitive inhibitor of the lysine methyltransferase SET8 (IC₅₀ = 7.3 µM; Kd = 18.3 µM). It is selective for SET8 over 15 other methyltransferases, including G9a and GLP (IC₅₀s = >100 µM).
Peptide sequence
N/A
CAS number
1620401-82-2
Molecular weight
413.56
Category
Biochemicals
Other name
6,7-dimethoxy-2-(pyrrolidin-1-yl)-N-(5-(pyrrolidin-1-yl)pentyl)quinazolin-4-amine
Molecular formula
C₂₃H₃₅N₅O₂
Physical appearance
Crystalline solid
Supplied with
N/A
Is this a salt?
No
Is it cell-permeable?
Yes
Purification
≥98% by HPLC
Reconstitute instructions
DMSO (~20 mg/ml)
Storage condition
-20°C
Shipping condition
gel pack
Maximum time for storage
36 months
Storage instructions
Protect from air and light
Tissue
cell
Additional description
For cells, cell lines and tissues in culture till half confluency.
