CGI-1746 for cell activation
Catalog number
9647-25
Name
CGI-1746 for cell activation
Size
25 mg
Price
545.00 EUR
Supplier
Details
Description
CGI-1746 is a potent, cell-permeable, ATP-competitive BTK inhibitor (IC₅₀ = 1.9 nM). It is specific for BTK, with around 1000-fold selectivity over Tec and Src family kinases.
Peptide sequence
N/A
CAS number
910232-84-7
Molecular weight
579.69
Category
Biochemicals
Other name
4-tert-butyl-N-[2-methyl-3-[4-methyl-6-[4-(morpholine-4-carbonyl)anilino]-5-oxopyrazin-2-yl]phenyl]benzamide
Molecular formula
C₃₄H₃₇N₅O₄
Physical appearance
Crystalline solid
Supplied with
N/A
Is this a salt?
No
Is it cell-permeable?
Yes
Purification
≥98% by HPLC
Reconstitute instructions
DMSO (>10 mg/ml)
Storage condition
-20°C
Shipping condition
gel pack
Maximum time for storage
36 months
Storage instructions
Protect from air and light
Tissue
cell
Additional description
For cells, cell lines and tissues in culture till half confluency.
