GSK-121 trifluoroacetate for cell activation
Catalog number
B1034-1000
Name
GSK-121 trifluoroacetate for cell activation
Size
1 mg
Price
186.00 EUR
Supplier
Details
Description
GSK-121 is a novel protein arginine deiminase 4 (PAD4) inhibitor. GSK-121 was shown to inhibit the citrullination of PAD4 target proteins in a functional assay with an IC₅₀ value of 3.2 µM.
Peptide sequence
N/A
CAS number
1652591-80-4
Molecular weight
501.5
Category
Biochemicals
Other name
(3-amino-1-piperidinyl)[1-methyl-2-(1-methyl-1H-indol-2-yl)-1H-benzimidazol-5-yl]-methanone, 2,2,2-trifluoroacetate
Molecular formula
C₂₃H₂₅N₅O •CF₃COOH
Physical appearance
Crystalline solid
Supplied with
N/A
Is this a salt?
No
Is it cell-permeable?
Yes
Purification
≥98%
Reconstitute instructions
DMSO (~30 mg/ml)
Storage condition
-20°C
Shipping condition
gel pack
Maximum time for storage
36 months
Storage instructions
Protect from air and moisture
Tissue
cell
Additional description
For cells, cell lines and tissues in culture till half confluency.
