CP-544326 for cell activation
Catalog number
B1121-5
Name
CP-544326 for cell activation
Size
5 mg
Price
175.00 EUR
Supplier
Details
Description
CP-544326 is a potent selective prostaglandin EP (2) receptor agonist which is the active acid metabolite of the prodrug PF-04217329 (Taprenepag isopropyl). CP-544326 was found to be a potent and selective EP(2) agonist (IC(₅₀) = 10 nM; EC(₅₀) = 2.8 nM) whose corneal permeability and ocular bioavailability are significantly increased when the compound is dosed as the isopropyl ester prodrug, PF-04217329.
Peptide sequence
N/A
CAS number
752187-80-7
Molecular weight
478.52
Category
Biochemicals
Other name
2-(3-((N-(4-(1H-pyrazol-1-yl)benzyl)pyridine-3-sulfonamido)methyl)phenoxy)acetic acid; Taprenepag
Molecular formula
C₂₄H₂₂N₄O₅S
Physical appearance
Crystalline solid
Supplied with
N/A
Is this a salt?
No
Is it cell-permeable?
Yes
Purification
≥98% by HPLC
Reconstitute instructions
DMSO (>10 mg/ml)
Storage condition
-20°C
Shipping condition
gel pack
Maximum time for storage
36 months
Storage instructions
Protect from air and light
Tissue
cell
Additional description
For cells, cell lines and tissues in culture till half confluency.
