Orexin 2 Receptor Agonist for cell activation

Orexin-2 receptor agonist is a potent and selective selective nonpeptidic orexin2 receptor (OX2R) agonist (OX2R EC₅₀ = 0.023 μM).

N/A

1796565-52-0 

586.22

Biochemicals

4'-methoxy-N,N-dimethyl-3'-(N-(3-((2-(3-methylbenzamido)ethyl)amino)phenyl)sulfamoyl)-[1,1'-biphenyl]-3-carboxamide

C₃₂H₃₄N₄O₅S

Crystalline solid

N/A

No

Yes

≥98% by HPLC

DMSO (>5 mg/ml)

-20°C

gel pack

36 months

Protect from air and light

cell

For cells, cell lines and tissues in culture till half confluency.The receptors are ligand binding factors of type 1, 2 or 3 and protein-molecules that receive chemical-signals from outside a cell. When such chemical-signals couple or bind to a receptor, they cause some form of cellular/tissue-response, e.g. a change in the electrical-activity of a cell. In this sense, am olfactory receptor is a protein-molecule that recognizes and responds to endogenous-chemical signals, chemokinesor cytokines e.g. an acetylcholine-receptor recognizes and responds to its endogenous-ligand, acetylcholine. However, sometimes in pharmacology, the term is also used to include other proteins that are drug-targets, such as enzymes, transporters and ion-channels.