CPI-0610 for cell activation
Catalog number
B1201-5
Name
CPI-0610 for cell activation
Size
5 mg
Price
186.00 EUR
Supplier
Details
Description
CPI-0610 is a potent, selective BET (bromodomain and extra terminal family of proteins) inhibitor and inhibits BRD4-BD1 with IC₅₀ of 39 nM. It potentially demonstrates anti-neoplastic activity by binding acetylated lysine recognition motifs on the bromodomain of BET proteins, thus preventing the interaction of BET proteins and acetylated histone peptides.
Peptide sequence
N/A
CAS number
1380087-89-7
Molecular weight
365.82
Category
Biochemicals
Other name
(S)-2-(6-(4-chlorophenyl)-1-methyl-4H-benzo[c]isoxazolo[4,5-e]azepin-4-yl)acetamide
Molecular formula
C₂₀H₁₆ClN₃O₂
Physical appearance
White Solid
Supplied with
N/A
Is this a salt?
No
Is it cell-permeable?
Yes
Purification
≥98% by HPLC
Reconstitute instructions
DMSO(>3 mg/ml)
Storage condition
-20°C
Shipping condition
gel pack
Maximum time for storage
36 months
Storage instructions
Protect from air and light
Tissue
cell
Additional description
For cells, cell lines and tissues in culture till half confluency.
