HDAC6 Inhibitor Screening Kit (Fluorometric)

-80°C

High-throughput compatible, quick and easy screening for HDAC6 ligands; Includes human recombinant HDAC6

dry ice

12 months

Human

• Rapid, high-throughput screening of drugs and novel ligands. • Development of structure-activity relationship (SAR) models to predict HDAC6 interaction liability of novel compounds.

Samples containing drugs, inhibitors or ligands (compounds that can interact and affect HDAC6 activity)

Tissue, pathway, proteinase, peptidase, protease ,acrosin, lipoprotein, activator, caspase, trypsin, papain, esterase inhibitors are proteins or receptor ligands or receptor antagonists that bind to an enzyme receptor and decreases its activity. Since blocking an enzyme's activity can kill a pathogen or correct a metabolic imbalance, many drugs are enzyme inhibitors. Not all receptor antagonist that bind to enzymes are inhibitors; enzyme activator ligands or agonists bind to enzymes and increase their enzymatic activity, while enzyme substrates bind and are converted to products in the normal catalytic cycle of the enzyme.