Renin Inhibitor

Aliskiren Hemifumarate; (2S,4S,5S,7S)-N-(2-Carbamoyl-2-methylpropyl)-5-amino-4-hydroxy-2,7-diisopropyl-8-[4-methoxy-3-(3-methoxypropoxy)phenyl]-octanamide hemifumarate

Crystalline solid

N/A

173334-58-2

N/A

C₃₀H₅₃N₃O₆ • ½C₄H₄O₄

609.79

≥98%

DMSO (>100 mg/ml) or H2O (>100 mg/ml)

Protect from moisture

A potent renin inhibitor

-20°C

gel pack

24 months

MFCD10566724

9939627

Biochemicals

Tissue, pathway, proteinase, peptidase, protease ,acrosin, lipoprotein, activator, caspase, trypsin, papain, esterase inhibitors are proteins or receptor ligands or receptor antagonists that bind to an enzyme receptor and decreases its activity. Since blocking an enzyme's activity can kill a pathogen or correct a metabolic imbalance, many drugs are enzyme inhibitors. Not all receptor antagonist that bind to enzymes are inhibitors; enzyme activator ligands or agonists bind to enzymes and increase their enzymatic activity, while enzyme substrates bind and are converted to products in the normal catalytic cycle of the enzyme.