PF-04981517 for cell activation

Catalog number
2917-5
Name
PF-04981517 for cell activation
Size
5 mg
Price
164.00 EUR
Supplier

Details

Description
Potent and selective inhibitor of CYP3A (IC50 = 30 nM (CYP3A4), 17 μM (CYP3A5) and 70 μM (CYP3A7).
Peptide sequence
N/A
CAS number
1390637-82-7
Molecular weight
456.6
Category
CYP inhibitor,Biochemicals
Other name
1-methyl-3-[1-methyl-5-(4-methylphenyl)-1H-pyrazol-4-yl]-4-[(3S)-3-(1-piperidinyl)-1-pyrrolidinyl]-1H-pyrazolo[3,4-d]pyrimidine, CYP3cide
Molecular formula
C₂₆H₃₂N₈
Physical appearance
Crystalline solid
Supplied with
N/A
Is this a salt?
No
Is it cell-permeable?
Yes
Purification
≥98%
Reconstitute instructions
DMSO (~20 mg/ml), DMF (~30 mg/ml), Ethanol (~2 mg/ml)
Storage condition
-20°C
Shipping condition
gel pack
Maximum time for storage
24 months
Storage instructions
Protect from air, light and moisture
Tissue
cell
Additional description
For cells, cell lines and tissues in culture till half confluency.