Bromodomain Inhibitor, (+)-JQ1

Catalog number
2070-5
Name
Bromodomain Inhibitor, (+)-JQ1
Size
5 mg
Price
555.00 EUR
Supplier

Details

Alternate Name/Synonyms
t-Butyl-2-((6S)-4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)acetate
Appearance
Off-white solid
Formulation
N/A
CAS Number
1268524-70-4
Peptide sequence
N/A
Molecular Formula
C₂₃H₂₅ClN₄O₂S
Molecular Weight
456.99
Purity
≥98% by HPLC
Solubility/Reconstitution Instructions
DMSO (10 mM)
Handling
Protect from air and moisture
Tagline
A potent and highly specific BET inhibitor
Storage Temp.
-20°C
Shipping Conditions
gel pack
Shelf Life
24 months
MDL Number
MFCD19443648
PubChem CID
46907787
Category
Biochemicals
Description
Tissue, pathway, proteinase, peptidase, protease ,acrosin, lipoprotein, activator, caspase, trypsin, papain, esterase inhibitors are proteins or receptor ligands or receptor antagonists that bind to an enzyme receptor and decreases its activity. Since blocking an enzyme's activity can kill a pathogen or correct a metabolic imbalance, many drugs are enzyme inhibitors. Not all receptor antagonist that bind to enzymes are inhibitors; enzyme activator ligands or agonists bind to enzymes and increase their enzymatic activity, while enzyme substrates bind and are converted to products in the normal catalytic cycle of the enzyme.