FAAH Inhibitor, PF-622 for cell activation

Catalog number
1928-25
Name
FAAH Inhibitor, PF-622 for cell activation
Size
25 mg
Price
480.00 EUR
Supplier

Details

Description
Cell-permeable. A potent and irreversible FAAH (Fatty Acid Amide Hydrolase) inhibitor. Inhibits FAAH in a time-dependent manner by covalently modifying the enzyme's active site serine (IC₅₀ = 33 nM). It is highly selective for FAAH relative to other mammalian serine hydrolases.
Peptide sequence
N/A
CAS number
898235-65-9
Molecular weight
346.43
Category
Biochemicals
Other name
N-Phenyl-4-(quinolin-2-ylmethyl)piperazine-1-carboxamide
Molecular formula
C₂₁H₂₂N₄O
Physical appearance
White soild
Supplied with
N/A
Is this a salt?
No
Is it cell-permeable?
Yes
Purification
≥98% by TLC
Reconstitute instructions
DMSO (~25 mg/ml) or Ethanol (~ 3 mg/ml)
Storage condition
-20°C
Shipping condition
gel pack
Maximum time for storage
36 months
Storage instructions
Protect from light and air
Tissue
cell
Additional description
For cells, cell lines and tissues in culture till half confluency.Tissue, pathway, proteinase, peptidase, protease ,acrosin, lipoprotein, activator, caspase, trypsin, papain, esterase inhibitors are proteins or receptor ligands or receptor antagonists that bind to an enzyme receptor and decreases its activity. Since blocking an enzyme's activity can kill a pathogen or correct a metabolic imbalance, many drugs are enzyme inhibitors. Not all receptor antagonist that bind to enzymes are inhibitors; enzyme activator ligands or agonists bind to enzymes and increase their enzymatic activity, while enzyme substrates bind and are converted to products in the normal catalytic cycle of the enzyme.