BAG 956 for cell activation

Catalog number
2456-25
Name
BAG 956 for cell activation
Size
25 mg
Price
567.00 EUR
Supplier

Details

Description
A potent, ATP-competitive, dual PI3K/PDK-1 inhibitor in vitro and in vivo (IC₅₀ = 56, 444, 34, 117 and 240 nM for PI3K p110-α ,β,d, γ, and PDK1 kinases, respectively). Displays anticancer properties.
Peptide sequence
N/A
CAS number
853910-02-8
Molecular weight
427.5
Category
Biochemicals
Other name
α,α,-Dimethyl-4-[2-methyl-8-[2-(3-pyr​idinyl)ethynyl]-1H-imidazo[4,5-c]quinolin-1-yl]-be​nzeneacetonitrile
Molecular formula
C₂₈H₂₁N₅
Physical appearance
Red solid
Supplied with
N/A
Is this a salt?
No
Is it cell-permeable?
Yes
Purification
≥98% by HPLC
Reconstitute instructions
DMSO (~15 mg/ml) or EtOH (~7 mg/ml)
Storage condition
-20°C
Shipping condition
gel pack
Maximum time for storage
24 months
Storage instructions
Protect from air and light
Tissue
cell
Additional description
For cells, cell lines and tissues in culture till half confluency.