GSK-1059615 for cell activation

Catalog number
9450-5
Name
GSK-1059615 for cell activation
Size
5 mg
Price
175.00 EUR
Supplier

Details

Description
GSK-1059615 is a potent, reversible, ATP-competitive inhibitor of PI3Kα (IC₅₀ = 2 nM). It inhibits proliferation in BT474 cells and attenuates MAPK signaling.
Peptide sequence
N/A
CAS number
958852-01-2
Molecular weight
333.36
Category
Biochemicals
Other name
5Z-​[[4-​(4-​pyridinyl)-​6-​quinolinyl]methylene]-​2,​4-​thiazolidinedione
Molecular formula
C₁₈H₁₁N₃O₂S
Physical appearance
Off-white solid
Supplied with
N/A
Is this a salt?
N/A
Is it cell-permeable?
Yes
Purification
≥98% by HPLC
Reconstitute instructions
DMSO (~4 mg/ml)
Storage condition
-20°C
Shipping condition
Gel pack
Maximum time for storage
36 months
Storage instructions
Protect from air and light
Tissue
cell
Additional description
For cells, cell lines and tissues in culture till half confluency.