C646, p300/CBP Inhibitor

Catalog number
1948-5
Name
C646, p300/CBP Inhibitor
Size
5 mg
Price
505.00 EUR
Supplier

Details

Alternate Name/Synonyms
(E)-4-(4-((5-(4,5-Dimethyl-2-nitrophenyl)furan-2-yl)-methylene)-3-methyl-5-oxo-4,5-dihydro-1H-pyrazol-1-yl)benzoic acid
Appearance
Red solid
Formulation
N/A
CAS Number
328968-36-1
Peptide sequence
N/A
Molecular Formula
C₂₄H₁₉N₃O₆
Molecular Weight
445.42
Purity
≥98% by NMR
Solubility/Reconstitution Instructions
DMSO (25 mM)
Handling
Protect from light and air
Tagline
A reversible, p300/CBP (CREB-binding protein) histone acetyltransferase (HAT) inhibitor
Storage Temp.
-20°C
Shipping Conditions
gel pack
Shelf Life
36 months
MDL Number
MFCD01784780
PubChem CID
1285941
Category
Biochemicals
Description
Tissue, pathway, proteinase, peptidase, protease ,acrosin, lipoprotein, activator, caspase, trypsin, papain, esterase inhibitors are proteins or receptor ligands or receptor antagonists that bind to an enzyme receptor and decreases its activity. Since blocking an enzyme's activity can kill a pathogen or correct a metabolic imbalance, many drugs are enzyme inhibitors. Not all receptor antagonist that bind to enzymes are inhibitors; enzyme activator ligands or agonists bind to enzymes and increase their enzymatic activity, while enzyme substrates bind and are converted to products in the normal catalytic cycle of the enzyme.